Browse Target: Ion Channel Category: Ligand-gated ion channel

Target ID Target Name Target Organism # Natural Product # Activity Record
NPT1530 Serotonin (5-HT) receptor Rattus norvegicus 20 31
NPT1783 Serotonin 3 (5-HT3) receptor Homo sapiens 6 7
NPT2959 Serotonin 3 (5-HT3) receptor Rattus norvegicus 2 9
NPT425 Serotonin 3a (5-HT3a) receptor Homo sapiens 13 18
NPT5252 Serotonin 3a (5-HT3a) receptor Rattus norvegicus 1 1
NPT5253 Serotonin 3 receptor (5HT3) Mus musculus 1 1
NPT5258 Serotonin 3a (5-HT3a) receptor Mus musculus 1 1
NPT473 Amiloride-sensitive sodium channel, ENaC Homo sapiens 1 1
NPT1000 GABA-A receptor; alpha-2/beta-3/gamma-2 Homo sapiens 4 13
NPT1001 GABA-A receptor; alpha-3/beta-3/gamma-2 Homo sapiens 4 12
NPT1002 GABA A receptor alpha-4/beta-3/gamma-2 Homo sapiens 4 4
NPT1003 GABA-A receptor; alpha-5/beta-3/gamma-2 Homo sapiens 4 11
NPT1004 GABA-A receptor; alpha-6/beta-3/gamma-2 Homo sapiens 5 5
NPT1007 GABA-A receptor; alpha-1/beta-2/gamma-2 Homo sapiens 16 37
NPT1008 GABA receptor rho-1 subunit Homo sapiens 6 14
NPT1009 GABA A receptor alpha-2/beta-2/gamma-2 Homo sapiens 3 7
NPT1010 GABA A receptor alpha-3/beta-2/gamma-2 Homo sapiens 4 9
NPT1324 GABA receptor rho-2 subunit Homo sapiens 1 1
NPT1325 GABA-A receptor; anion channel Bos taurus 5 15
NPT1326 GABA-A receptor; anion channel Mus musculus 5 10
NPT1402 GABA receptor alpha-2 subunit Rattus norvegicus 2 4
NPT1404 GABA receptor gamma-1 subunit Rattus norvegicus 3 3
NPT1406 GABA receptor alpha-1 subunit Homo sapiens 1 2
NPT1408 GABA-A receptor; agonist GABA site Homo sapiens 3 6
NPT1409 GABA receptor alpha-6 subunit Rattus norvegicus 1 1
NPT1410 GABA receptor alpha-1 subunit Rattus norvegicus 2 4
NPT1411 GABA receptor alpha-3 subunit Rattus norvegicus 1 1
NPT1412 GABA receptor alpha-4 subunit Rattus norvegicus 1 1
NPT1413 GABA receptor alpha-5 subunit Rattus norvegicus 2 2
NPT2643 GABA-A receptor; GABA-A site (alpha1/beta2 interface) Homo sapiens 3 6
NPT5809 GABA A receptor alpha-1/beta-1/gamma-2 Homo sapiens 1 1
NPT5810 GABA receptor beta-3 subunit Homo sapiens 1 1
NPT6132 GABA A receptor alpha-3/beta-2/gamma-2 Rattus norvegicus 1 4
NPT6133 GABA A receptor alpha-6/beta-2/gamma-2 Rattus norvegicus 1 6
NPT6134 GABA A receptor alpha-6/beta-2/gamma-2 Homo sapiens 1 2
NPT6135 GABA A receptor alpha-2/beta-2/gamma-2 Rattus norvegicus 1 1
NPT6136 GABA A receptor alpha-5/beta-3/gamma-2 Rattus norvegicus 1 1
NPT6140 GABA receptor alpha-2 subunit Homo sapiens 1 1
NPT6141 GABA receptor alpha-3 subunit Homo sapiens 1 1
NPT6142 GABA receptor alpha-5 subunit Homo sapiens 1 2
NPT735 GABA receptor subunit Musca domestica 22 22
NPT805 GABA-A receptor; anion channel Rattus norvegicus 62 184
NPT899 GABA-A receptor; alpha-1/beta-2/gamma-2 Rattus norvegicus 8 52
NPT996 GABA-A receptor; anion channel Homo sapiens 20 37
NPT998 GABA-C receptor Homo sapiens 5 5
NPT999 GABA-A receptor; alpha-1/beta-3/gamma-2 Homo sapiens 7 13
NPT250 Glycine receptor Rattus norvegicus 2 4
NPT426 Glycine receptor subunit alpha-1 Homo sapiens 10 27
NPT4324 Glycine receptor subunit alpha-2 Homo sapiens 4 7
NPT4641 Glycine receptor subunit alpha-3 Homo sapiens 6 6
NPT3520 Inositol 1,4,5-trisphosphate receptor type 3 Bos taurus 1 1
NPT3522 Inositol 1,4,5-trisphosphate receptor type 1 Homo sapiens 1 2
NPT3523 Inositol 1,4,5-trisphosphate receptor Homo sapiens 1 4
NPT3524 Type 1 InsP3 receptor isoform S2 Sus scrofa 1 1
NPT3529 Inositol 1,4,5-trisphosphate receptor type 3 Homo sapiens 4 4
NPT3530 Inositol 1,4,5-trisphosphate receptor type 1 Rattus norvegicus 1 13
NPT1304 Nicotinic acetylcholine receptor alpha 5 subunit Musca domestica 11 14
NPT436 Nicotinic acetylcholine receptor alpha8 subunit Periplaneta americana 1 1
NPT2654 P2X purinoceptor 7 Homo sapiens 6 6
NPT2669 P2X purinoceptor 1 Rattus norvegicus 1 1
NPT2670 P2X purinoceptor 2 Homo sapiens 3 3
NPT2671 P2X purinoceptor 4 Rattus norvegicus 3 4
NPT2674 P2X purinoceptor 1 Homo sapiens 4 5
NPT2675 P2X purinoceptor 3 Homo sapiens 4 4
NPT2676 P2X purinoceptor 1 Mus musculus 1 1
NPT4494 P2X purinoceptor 5 Rattus norvegicus 2 2
NPT4495 P2X purinoceptor 6 Rattus norvegicus 2 2
NPT4953 P2X purinoceptor 2 Rattus norvegicus 1 1
NPT4954 P2X purinoceptor 4 Homo sapiens 2 3
NPT6603 P2X purinoceptor 7 Rattus norvegicus 1 1
NPT2699 Ryanodine receptor 1 Oryctolagus cuniculus 6 8
NPT2700 Ryanodine receptor 3 Mus musculus 1 1
NPT4277 Ryanodine receptor 1 Homo sapiens 5 6
NPT5115 Ryanodien receptor Spodoptera exigua 2 5
NPT3739 Glutamate receptor ionotropic, AMPA Rattus norvegicus 9 25
NPT3741 Glutamate receptor ionotropic, AMPA 1 Homo sapiens 3 14
NPT3742 Glutamate receptor ionotropic, AMPA 2 Homo sapiens 4 14
NPT3743 Glutamate receptor ionotropic, AMPA 4 Homo sapiens 4 10
NPT3750 Glutamate receptor ionotropic, AMPA 1 Rattus norvegicus 5 18
NPT3751 Glutamate receptor ionotropic, AMPA 2 Rattus norvegicus 3 16
NPT3752 Glutamate receptor ionotropic, AMPA 3 Rattus norvegicus 3 17
NPT3753 Glutamate receptor ionotropic, AMPA 4 Rattus norvegicus 3 13
NPT3758 Glutamate receptor ionotropic, AMPA 3 Homo sapiens 2 5
NPT5636 Glutamate receptor ionotropic, AMPA Mus musculus 1 1
NPT3737 Glutamate receptor ionotropic kainate 2 Homo sapiens 2 9
NPT3738 Glutamate receptor ionotropic kainate 2 Rattus norvegicus 4 22
NPT3740 Glutamate receptor ionotropic, kainate Rattus norvegicus 7 25
NPT3744 Glutamate receptor ionotropic kainate 1 Homo sapiens 2 9
NPT3745 Glutamate receptor ionotropic kainate 5 Homo sapiens 3 7
NPT3746 Glutamate receptor ionotropic kainate 3 Homo sapiens 2 4
NPT3748 Glutamate receptor ionotropic kainate 1 Rattus norvegicus 4 20
NPT3754 Glutamate receptor ionotropic kainate 4 Rattus norvegicus 1 1
NPT3755 Glutamate receptor ionotropic kainate 5 Rattus norvegicus 1 1
NPT3756 Glutamate receptor ionotropic kainate 3 Rattus norvegicus 3 8
NPT3920 Neuronal acetylcholine receptor; alpha4/beta4 Homo sapiens 2 6
NPT3921 Neuronal acetylcholine receptor; alpha2/beta4 Homo sapiens 3 4
NPT3924 Neuronal acetylcholine receptor protein alpha-4 subunit Rattus norvegicus 5 21
NPT3925 Acetylcholine receptor protein alpha chain Torpedo californica 6 10
NPT409 Neuronal acetylcholine receptor; alpha4/beta2 Homo sapiens 20 112
NPT410 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens 20 79
NPT411 Neuronal acetylcholine receptor; alpha3/beta4 Homo sapiens 12 56
NPT414 Neuronal acetylcholine receptor protein alpha-7 subunit Rattus norvegicus 13 91
NPT421 Neuronal acetylcholine receptor protein alpha-7 subunit Mus musculus 1 2
NPT423 Neuronal acetylcholine receptor; alpha3/beta2 Homo sapiens 6 11
NPT424 Neuronal acetylcholine receptor subunit alpha-3 Homo sapiens 3 10
NPT428 Neuronal acetylcholine receptor subunit alpha-3 Rattus norvegicus 5 12
NPT429 Neuronal acetylcholine receptor protein alpha-4 subunit Homo sapiens 3 6
NPT5028 Nicotinic acetylcholine receptor alpha3/betaX Homo sapiens 1 1
NPT5029 Neuronal acetylcholine receptor protein alpha-9 subunit Rattus norvegicus 1 2
NPT5033 Acetylcholine receptor protein alpha chain Homo sapiens 2 3
NPT5036 Neuronal acetylcholine receptor protein alpha-2 subunit Rattus norvegicus 2 6
NPT5037 Neuronal acetylcholine receptors; alpha-3/beta-4, alpha-5, beta-2 Homo sapiens 1 1
NPT5038 Neuronal acetylcholine receptor; alpha2/beta2 Homo sapiens 1 1
NPT5039 Neuronal acetylcholine receptor protein alpha-4 subunit Mus musculus 2 2
NPT5040 Neuronal acetylcholine receptor; alpha3/alpha6/beta2/beta3 Homo sapiens 1 2
NPT6604 Neuronal acetylcholine receptor protein alpha-10 subunit Rattus norvegicus 1 1
NPT3042 Neuronal nicotinic acetylcholine receptor Mus musculus 2 3
NPT3923 Neuronal acetylcholine receptor; alpha2/beta4 Rattus norvegicus 3 17
NPT412 Neuronal acetylcholine receptor; alpha4/beta2 Rattus norvegicus 18 169
NPT413 Neuronal acetylcholine receptor Rattus norvegicus 23 84
NPT415 Neuronal acetylcholine receptor; alpha2/beta2 Rattus norvegicus 5 22
NPT416 Neuronal acetylcholine receptor; alpha3/beta2 Rattus norvegicus 6 25
NPT417 Neuronal acetylcholine receptor; alpha3/beta4 Rattus norvegicus 9 62
NPT418 Neuronal acetylcholine receptor; alpha4/beta4 Rattus norvegicus 9 36
NPT4533 Acetylcholine receptor subunit beta-like 2 Drosophila melanogaster 3 5
NPT5031 Nicotinic acetylcholine receptor alpha2/beta4 Homo sapiens 1 1
NPT5035 Neuronal acetylcholine receptor subunit beta-4 Rattus norvegicus 2 2
NPT964 Nicotinic acetylcholine receptor alpha-4/beta-2 Mus musculus 4 4
NPT3919 Acetylcholine receptor; alpha1/beta1/delta/gamma Homo sapiens 3 8
NPT3922 Acetylcholine receptor Torpedo californica 13 19
NPT408 Acetylcholine receptor protein delta chain Torpedo californica 4 5
NPT5032 Muscle-type nicotinic acetylcholine receptor Homo sapiens 1 1
NPT6226 Acetylcholine receptor protein epsilon chain Homo sapiens 2 2
NPT1163 Glutamate (NMDA) receptor subunit zeta 1 Rattus norvegicus 15 21
NPT1496 Glutamate NMDA receptor Rattus norvegicus 24 65
NPT1837 Glutamate NMDA receptor; Grin1/Grin2a Rattus norvegicus 5 6
NPT1838 Glutamate NMDA receptor; Grin1/Grin2b Rattus norvegicus 3 4
NPT1839 Glutamate NMDA receptor; Grin1/Grin2c Rattus norvegicus 3 4
NPT3929 Glutamate NMDA receptor; GRIN1/GRIN2A Homo sapiens 3 4
NPT3930 Glutamate NMDA receptor; GRIN1/GRIN2B Homo sapiens 2 11
NPT3933 Glutamate [NMDA] receptor subunit epsilon 2 Rattus norvegicus 2 10
NPT4202 Glutamate [NMDA] receptor subunit epsilon 3 Rattus norvegicus 2 3
NPT4568 Glutamate receptors; NMDA/AMPA Rattus norvegicus 1 1
NPT5060 Ionotropic glutamate receptor NMDA 1/2D Rattus norvegicus 1 2
NPT5858 Glutamate [NMDA] receptor subunit epsilon 2 Mus musculus 1 2
NPT5859 Glutamate [NMDA] receptor subunit epsilon 2 Homo sapiens 1 2